interaction of a pharmaceutical water-soluble polymer with bio-relevant surfactants

DOI

We have been developing hydroxypropylmethyl cellulose (HPMC) microspheres for delivering poorly water-soluble drugs. The in vitro dissolution data showed that the presence of SDS is essential for obtaining a high level of drug release. The higher the level of drug that is released from the formulations, the greater the absorption and bioavailability of the formulation. Previous SANS data revealed some detail of the structure of the polymer-SDS complex and we have shown it is reasonable to hypothesise that the drug molecules may be encapsulated into the polymer-surfactant complex which leads to the improved dissolution of the poorly water-soluble model drug. Therefore the objectives of this proposed study are to investigate the influence of drug incorporation on the structure of the polymer-surfactant complex, and to expand the range of concentrations studied.

Identifier
DOI https://doi.org/10.5286/ISIS.E.24079869
Metadata Access https://icatisis.esc.rl.ac.uk/oaipmh/request?verb=GetRecord&metadataPrefix=oai_datacite&identifier=oai:icatisis.esc.rl.ac.uk:inv/24079869
Provenance
Creator Dr Stephen Roser; Professor Karen Edler
Publisher ISIS Neutron and Muon Source
Publication Year 2013
Rights CC-BY Attribution 4.0 International; https://creativecommons.org/licenses/by/4.0/
OpenAccess true
Contact isisdata(at)stfc.ac.uk
Representation
Resource Type Dataset
Discipline Photon- and Neutron Geosciences
Temporal Coverage Begin 2010-05-04T08:32:57Z
Temporal Coverage End 2010-05-06T09:28:49Z