Effect of protein lipidation on adsorption and surface-associated protein fibrillation

DOI

Lipidation of proteins is used in the pharmaceutical industry to improve the therapeutic efficacy of proteins. However, there is a limited knowledge on the physicochemical properties of these lipidated proteins. They may form irreversible multilayers upon adsorption onto solid surfaces, which in turn may catalyze the formation of surface-associated protein fibrillation. Fibrillation of proteins is considered to be a cause of multiple serious diseases. Insulin detemir, a human insulin analogue, with a fatty acid chain attached to the protein, was used as model compound, and compared to human insulin. Initial AFM and QCM-D results have shown that the lipid chain significant increases the initial adsorption and subsequent formation of fibrils onto hydrophobic surfaces. NR data can give a unique structural insight into the initial adsorbed (multi)-layers, density and thickness of these layers as well as for surface-associated fibrils. This structural insight will be of great significance in exploiting lipidation of proteins as a safe method to improve the therapeutic activity of proteins and understand the impact of the lipid chain in the adsorption process and subsequent fibrillation.

Identifier
DOI https://doi.org/10.5291/ILL-DATA.8-02-711
Metadata Access https://data.ill.fr/openaire/oai?verb=GetRecord&metadataPrefix=oai_datacite&identifier=10.5291/ILL-DATA.8-02-711
Provenance
Creator Browning, Kathryn; Cardenas, Marite; Nordstrom, Randi; Campbell, Richard; Maric, Selma; Hedegaard, Sofie; Lind, Tania
Publisher Institut Laue-Langevin
Publication Year 2016
Rights OpenAccess; info:eu-repo/semantics/openAccess
OpenAccess true
Representation
Resource Type Dataset
Size 2 GB
Version 1
Discipline Particles, Nuclei and Fields