GLUTATHIONE-MEDIATED RESISTANCE TO Pt- AND Pd-BASED ANTICANCER DRUGS PROBED BY SIMULTANEOUS INS AND RAMAN SCATTERING

DOI

The present study aims at using simultaneous INS and Raman scattering experiments to elucidate resistance to cisplatin-like Pt(II)- and Pd(II)-based anticancer agents via glutathione detoxification. Drug binding to this endogenous sulfur-containing tripeptide will be investigated, as compared to the major pharmacological target (DNA). Apart from cisplatin, the mono- and polynuclear complexes Pt(dap)Cl2 and Pt2(Spm)Cl4 will be studied, as well as their Pd(II) counterparts. The results thus obtained will be analysed in the light of previously obtained INS and theoretical data for these compounds and for cisplatin´s interplay with DNA, as well as for glutathione competition towards cisplatin-DNA adducts.

Identifier
DOI https://doi.org/10.5286/ISIS.E.42578971
Metadata Access https://icatisis.esc.rl.ac.uk/oaipmh/request?verb=GetRecord&metadataPrefix=oai_datacite&identifier=oai:icatisis.esc.rl.ac.uk:inv/42578971
Provenance
Creator Dr Maria Paula Marques; Dr Ana Carvalho; Dr Luis Alberto Batista de Carvalho; Professor Stewart Parker
Publisher ISIS Neutron and Muon Source
Publication Year 2017
Rights CC-BY Attribution 4.0 International; https://creativecommons.org/licenses/by/4.0/
OpenAccess true
Contact isisdata(at)stfc.ac.uk
Representation
Resource Type Dataset
Discipline Biology; Biomaterials; Chemistry; Engineering Sciences; Life Sciences; Materials Science; Materials Science and Engineering; Medicine; Natural Sciences
Temporal Coverage Begin 2013-12-06T08:06:52Z
Temporal Coverage End 2014-02-17T10:05:55Z